| 货号 | 1175/100U |
| 是否允许进口 | 否 |
| 是否危险品 | 是 |
| 供应商 | Tocris |
| 生物活性 | Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 2516 |
| 分子式 | C103H147N27O |
| 可溶性/溶解性 | Soluble to 1 mg/ml in water |
| 序列号 | CTCNDMTDEECLNFCHQDVIW (Modifications: Disulfide bridge between 1 - 15, 3 - 11) |
| 参考文献 | Miasiroet al (1998) Distinct endothelin-B receptors mediate the effects of sarafotoxin S6c and IRL 1620 in the ileum. J.Cardiovasc.Pharmacol. 31 S175. PMID: 9595431. Matsuoet al (1997) Effects of sarafotoxin S6c on antidiuresis and norepinephrine overflow induced by stimulation of renal nerves in anesthetized dogs. J.Pharmacol.Exp.Ther. 280 905. PMID: 9023305. Williamset al (1993) Characterization of cloned human endothelin receptors. Life Sci. 53 407. PMID: 8336519. Williamset al (1991) Sarafotoxin S6c: an agonist which distinguishes between endothelin receptor subtypes. Biochem.Biophys.Res.Commun. 175 556. PMID: 1850245. |