| 货号 | 1899/100U |
| 是否允许进口 | 否 |
| 是否危险品 | 是 |
| 供应商 | Tocris |
| 生物活性 | Endothelin receptor agonist (EC50 values are 7.5 and > 150 nM for contraction of pig coronary artery and guinea pig aorta respectively). Nociceptive in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 2514.85 |
| 分子式 | C105H156N28O |
| 可溶性/溶解性 | Soluble to 1 mg/ml in water |
| 序列号 | CSCKDMTDKECLNFCHQDVIW (Modifications: Disulfide bridge between 1 - 15, 3 - 11) |
| 参考文献 | Raffaet al (1996) Endothelin-induced nociception in mice: mediation by ETA and ETB receptors. J.Pharmacol.Exp.Ther. 276 647. PMID: 8632332. Schoeffter and Randriantsoa (1993) Differences between endothelial receptors mediating contraction of guinea-pig aorta and pig coronary artery. Eur.J.Pharmacol. 249 199. PMID: 8287901. Minkeset al (1992) Comparison of responses to sarafotoxins 6a and 6c in pulmonary and systemic vascular beds. Am.J.Physiol. 262 H852. PMID: 1348398. |