6-Iodoresiniferatoxin (1 MG)
货号：
1556/1 基本售价：
询价 规格：
1 mg
产品信息
概述| 货号 | 1556/1 |
| 别名 | [(2S,3aR,3bS,6aR,9aR,9bR,10R,11aR)-3a,3b,6,6a,9a,10,11,11a-octahydro-6a-hydroxy-8,10-dimethyl-11a-(1-methylethenyl)-7-oxo-2-(phenylmethyl)-7H-2,9b-epoxyazuleno[5,4-e]-1,3-benzodioxol-5-yl]-4-hydroxy-2-iodo-5-methoxy-benzeneacetic acid methyl ester; 6'-IRTX |
| 是否允许进口 | 否 |
| 是否危险品 | 是 |
性能| 供应商 | Tocris |
| 生物活性 | High affinity TRPV1 (VR1) vanilloid receptor partial agonist (Ki = 0.71 nM; EC50 = 130 nM at human VR1). Displays partial agonism at human VR1 and full agonism at rat VR1. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >98 % |
| 计算分子量 | 754.6 |
| 分子式 | C37H39IO9 |
| 可溶性/溶解性 | Soluble in ethanol and in DMSO |
| 参考文献 | McDonnellet al (2002) Synthesis and in vitro evaluation of a novel iodinated resiniferatoxin derivative that is an agonist at the human vanilloid VR1 receptor. Bioorg.Med.Chem.Lett. 12 1189. PMID: 11934585. |
