| 货号 | 1362/1 |
| 别名 | 6,7-Deepoxy-6,7-didehydro-5-deoxy-2 |
| 是否允许进口 | 否 |
| 是否危险品 | 是 |
| 供应商 | Tocris |
| 生物活性 | Potent and silent vanilloid receptor antagonist, 40-fold more potent than capsazepine (Cat. No. 0464). Binds to TRPV1 (VR1) receptors expressed in HEK293 cells with a Ki of 5.8 nM. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >98 % |
| 计算分子量 | 754.6 |
| 分子式 | C37H39IO9 |
| 可溶性/溶解性 | Soluble in DMSO and to 100 mM in ethanol |
| 参考文献 | Marinelliet al (2002) Capsaicin activation of glutamatergic synaptic transmission in the rat locus coeruleus in vitro. J.Physiol. 543 531. PMID: 12205187. Seabrooket al (2001) Properties of iodo-resiniferatoxin - a high affinity VR1 vanilloid receptor antagonist. Soc.Neurosci.Abstr. 925.9. Wahlet al (2001) Iodo-resiniferatoxin, a new potent vanilloid receptor antagonist. Mol.Pharmacol. 59 9. PMID: 11125018. |