货号 | 0789/1 |
别名 | (±)-2-Acetyl-9-aza bicyclo[4.2.1]non-2-ene fumarate |
是否允许进口 | 否 |
是否危险品 | 是 |
供应商 | Tocris |
生物活性 | A potent nicotinic agonist (Ki values are 1.25 and 1840 nM for α4β2 and α7 nicotinic receptors respectively). Stimulates [3H]-dopamine release from rat striatal synaptosomes (EC50 = 136 nM). |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >96 % |
计算分子量 | 281.31 |
分子式 | C10H15NO.C4H |
可溶性/溶解性 | Soluble to 50 mM in water |
参考文献 | Sharpleset al (2000) UB-165 implicates α4β2 nAChR in striatal dopamine release. J.Neurosci. 20 2783. PMID: 10751429. Thomaset al (1993) (+)-Anatoxin is a potent agonist at neuronal nicotinic acetylcholine receptors. J.Neurochem. 60 2308. PMID: 8492133. Gordonet al (1992) Induced release of acetylcholine from guinea pig ileum longitudinal muscle myenteric plexus by anatoxin-A. J.Pharmacol.Exp.Ther. 263 997. PMID: 1469655. Stolermanet al (1992) Behavioural effects of anatoxin, a potent nicotinic agonist in rats. Neuropharmacology 31 311. PMID: 1630597. |