| 货号 | 1104/50 |
| 别名 | 1-[2-Chloro-6-[[(3-iodophenyl)methy |
| 供应商 | Tocris |
| 生物活性 | High affinity and extremely selective A3 adenosine receptor agonist (Ki = 0.33 nM). Displays 2500- and 1400-fold selectivity over A1 and A2A receptors respectively. Exhibits high selectivity over the Na+-independent adenosine transporter. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 544.74 |
| 分子式 | C18H18ClIN6O4 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| CAS号 | 163042-96-4 |
| 参考文献 | Jacobson (1998) Adenosine A3 receptors: novel ligands and paradoxical effects. TiPS 19 184. PMID: 9652191. Schaicket al (1996) Hemodynamic effects of histamine release elicited by the selective adenosine A3 receptor agonist 2-Cl-IB-MECA in conscious rats. Eur.J.Pharmacol. 308 311. PMID: 8858305. Kimet al (1994) 2-Substitution of N6-benzyladenosine-5'-uronamides enhances selectivity for A3 adenosine receptors. J.Med.Chem. 37 3614. PMID: 7932588. |