货号 | 1063/50 |
别名 | 4-[2-[[6-Amino-9-(N-ethyl-β-D-ribofu |
供应商 | Tocris |
生物活性 | A2A adenosine receptor agonist (Ki = 27 nM). Has affinity for A1 and A3 adenosine receptors but can be used to distinguish A2A- and A2B-mediated effects. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
纯度 | >98 % |
计算分子量 | 535.99 |
分子式 | C23H29N7O6.HCl |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
CAS号 | 124182-57-6 |
参考文献 | Klot (2000) Adenosine receptors and their ligands. Naunyn Schmiedebergs Arch.Pharmacol. 362 382. PMID: 11111832. Nekooeian and Tabrizchi (1998) Effects of CGS 21680, a selective A2A adenosine receptor agonist, on cardiac output and vascular resistance in acute heart failure in the anaesthetized rat. Br.J.Pharmacol. 123 1666. PMID: 9605574. Philliset al (1990) The selective adenosine A2 receptor agonist, CGS 21680, is a potent depressant of cerebral cortical neuronal activity. Brain Res. 509 328. PMID: 2322828. |