(+/-)-LY 395756 (50 MG)
货号:
3272/50 基本售价:
16438.2 元 规格:
50 mg
产品信息
概述货号 | 3272/50 |
别名 | (1S,2S,4R,5R,6S)-rel-2-Amino-4-methylbicyclo[3.1.0]hexane-2,6-dicarboxylic acid |
性能供应商 | Tocris |
生物活性 | Selective metabotropic glutamate ligand for mGlu2and mGlu3 receptors (Ki values are 0.165 μM and 0.302 μM respectively). Acts as an agonist at mGlu2 and antagonist at mGlu3. Analog of LY 354740 (Cat. No. 3246). |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >98 % |
计算分子量 | 199.21 |
分子式 | C9H13NO4 |
可溶性/溶解性 | Soluble to 100 mM in 1eq. HCl and to 100 mM in 1eq. NaOH |
CAS号 | 842679-66-4 |
参考文献 | Dominguezet al (2005) Methyl substitution of 2-aminobicyclo[3.1.0]hexane 2,6-dicarboxylate (LY354740) determines functional activity at metabotropic glutamate receptors: identification of a subtype selective mGlu2 receptor agonist. J.Med.Chem. 48 3605. PMID: 15887967. |