GP 2a (50 MG)
货号:
2678/50 基本售价:
13761.3 元 规格:
50 mg
产品信息
概述货号 | 2678/50 |
别名 | N-Cyclohexyl-1-(2,4-dichlorophenyl)-1,4-dihydro-6-methylindeno[1,2-c]pyrazole-3-carboxamide |
性能供应商 | Tocris |
生物活性 | Selective CB2 receptor agonist; Ki values are 7.6 and 900 nM for CB2 and CB1 receptors respectively. Increases P-ERK1/2 expression in HL-60 cells in vitro. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 440.36 |
分子式 | C24H23Cl2N3< |
可溶性/溶解性 | Soluble to 50 mM in DMSO and to 20 mM in ethanol |
参考文献 | Murinedduet al (2006) Tricyclic pyrazoles. 4. Synthesis and biological evaluation of analogues of the robust and selective CB2 cannabinoid ligand 1-(2',4'-dichlorophenyl)-6-methyl-N-piperidin-1-yl-1,4-dihydroindeno[1,2-c]pyrazole-3-carboxamide. J.Med.Chem. 49 7502. PMID: 17149879. |