货号 | 1242/50 |
别名 | N-[3-[3-(Dimethylamino)ethoxy]-4-me |
供应商 | Tocris |
生物活性 | A selective h5-HT1B antagonist with approximately 25-fold selectivity over h5-HT1D and little or no affinity for a range of other receptor types. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 523.03 |
分子式 | C28H30N4O4.HCl |
可溶性/溶解性 | Soluble to 50 mM in water |
CAS号 | 170230-39-4 |
参考文献 | Haganet al (1997) Stimulation of 5-HT1B receptors causes hypothermia in the guinea pig. Eur.J.Pharmacol. 331 169. PMID: 9274976. Priceet al (1997) SB-216641 and BRL-15572 - compounds to pharmacologically discriminate h5-HT1B and h5-HT1D receptors. Naunyn Schmiedebergs Arch.Pharmacol. 356 312. PMID: 930567. Schlickeret al (1997) Effects of selective h5-HT1B (SB-216641) and 5-HT1D (BRL-15572) receptor ligands on guinea pig and human 5-HT auto- and heteroreceptors. Naunyn Schmiedebergs Arch.Pharmacol. 356 321. PMID: 9303568. |