NNC 63-0532 (50 MG)
货号：
1780/50 基本售价：
13077.2 元 规格：
50 mg
产品信息
概述| 货号 | 1780/50 |
| 别名 | 8-(1-Naphthalenylmethyl)-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decane-3-acetic acid, methyl ester |
性能| 供应商 | Tocris |
| 生物活性 | Potent non-peptide agonist for the NOP receptor (EC50 = 305 nM, Ki = 7.3 nM); ~ 12-fold selective over other receptors. Centrally active following systemic administration in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 443.54 |
| 分子式 | C27H29N3O3 |
| 可溶性/溶解性 | Soluble to 5 mM in ethanol and to 50 mM in DMSO |
| CAS号 | 250685-44-0 |
| 参考文献 | Thomsen and Hohlweg (2000) (8-Naphthalen-1-ylmethyl-4-oxo-1-phenyl-1,3,8-triaza-spiro[4.5]-dec-3-yl)-acetic acid methyl ester (NNC 63-0532) is a novel potent nociceptin receptor agonist. Br.J.Pharmacol. 131 903. PMID: 11053209. |
