MA 2029 (50 MG)
货号：
4934/50 基本售价：
13077.2 元 规格：
50 mg
产品信息
概述| 货号 | 4934/50 |
| 别名 | 4-Fluoro-N-methyl-L-phenylalanyl-N-methyl-L-valyl-3-(1,1-dimethylethyl)-N-ethyl-L-tyrosinamide |
性能| 供应商 | Tocris |
| 生物活性 | Potent and selective, competitive motilin receptor antagonist (IC50 = 4.9 nM). Selective for the motilin receptor over a range of other receptors and ion channels. Inhibits motilin-induced duodenal muscle contractions in vitro. Also inhibits motilin-induced colonic and abdominal contractions in vivo. Orally active. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 556.71 |
| 分子式 | C31H45FN4O4< |
| 可溶性/溶解性 | Soluble to 20 mM in 1eq. HCl and to 100 mM in DMSO |
| 参考文献 | Sudoet al (2008) Oral administration of MA-2029, a novel selective and competitive motilin receptor antagonist, inhibits motilin-induced intestinal contractions and visceral pain in rabbits. Eur.J.Pharmacol. 581 296. PMID: 18164286. |
