TFM-4AS-1 (50 MG)
货号:
3813/50 基本售价:
12274.1 元 规格:
50 mg
产品信息
概述货号 | 3813/50 |
别名 | (1S,3aS,3bS,5aR,9aR,9bS,11aS)-6,9a,11a-Trimethyl-7-oxo-N-[2-(trifluoromethyl)phenyl]-2,3,3a,3b,4,5,5a,9b,10,11-decahydro-1H-indeno[5,4-f]quinoline-1-carboxamide |
性能供应商 | Tocris |
生物活性 | Potent selective androgen receptor modulator (SARM) (IC50 = 30 nM). Steroidal compound. Exhibits limited effects on reproductive tissues and sebaceous glands; does not repress AP-1-sensitive MMP-1 reporter. Inhibits 5α-reductase type I and II (IC50 values are 2 and 3 nM respectively). |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 474.56 |
分子式 | C27H33F3N2 |
可溶性/溶解性 | Soluble to 10 mM in DMSO and to 10 mM in ethanol |
参考文献 | Schmidtet al (2009) Identification of anabolic selective androgen receptor modulators with reduced activities in reproductive tissues and sebaceous glands. J.Biol.Chem. 284 36367. PMID: 19846549. |