| 货号 | 0764/50 |
| 别名 | (+)-4-[(αR)-α-((2S,5R)-4-Allyl-2,5-di |
| 供应商 | Tocris |
| 生物活性 | A highly selective and potent non-peptide δ-opioid agonist, 2000-fold selective over μ-opioid receptors. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 449.64 |
| 分子式 | C28H39N3O2 |
| 可溶性/溶解性 | Soluble to 100 mM in 1eq. HCl with gentle warming and to 20 mM in DMSO |
| CAS号 | 156727-74-1 |
| 参考文献 | Knappet al (1996) Structure-activity relationships for SNC80 and related compounds at cloned human deltaandmu opioid receptors. J.Pharmacol.Exp.Ther. 277 1284. PMID: 8667189. Bilskyet al (1995) SNC 80, a selective, nonpeptidic and systemically active opioid δ agonist. J.Pharmacol.Exp.Ther. 273 359. PMID: 7714789. Calderonet al (1994) Probes for narcotic receptor mediated phenomena. 19. Synthesis of (+)-4-[(αR)-α-((2S,5R)-4-allyl-2,5-dimethyl-1-piperazinyl)-3-methoxybenzyl]-N,N-diethylbenzamide (SNC80): a highly selective nonpeptide σ opioid receptor agonist. J.Med.Chem. 37 2125. PMID: 8035418. |