| 货号 | 2752/50 |
| 别名 | N-(4-Cyanophenyl)-2-[4-(2,3,6,7-tet |
| 供应商 | Tocris |
| 生物活性 | Selective adenosine A2B receptor antagonist (Ki values are 1.97, 16.8, 403, 503, 570 and 612 nM for hA2B, rA1, hA1, hA2A, hA3 and rA2A receptors respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 486.52 |
| 分子式 | C26H26N6O4 |
| 可溶性/溶解性 | Soluble to 5 mM in DMSO with gentle warming and to 10 mM in DMSO with sonication |
| CAS号 | 264622-58-4 |
| 参考文献 | Nemethet al (2007) Adenosine receptor activation ameliorates type I diabetes. FASEB J. 212380. Jiet al (2001) [3H]MRS 1754, a selective antagonist radioligand for A2B adenosine receptors. Biochem.Pharmacol. 61 657. PMID: 11266650. Kimet al (2000) Anilide derivatives of an 8-phenylxanthine carboxylic congener are highly potent and selective antagonists at human A2B adenosine receptors. J.Med.Chem. 43 1165. PMID: 10737749. |