货号 | 4163/50 |
别名 | N-(Cyclohexylmethyl)-2-[(5-[(phenyl |
供应商 | Tocris |
生物活性 | NMDA receptor antagonist, selective for NR1/NR2A (pIC50 = 5.4) over NR1/NR2B. |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >99 % |
计算分子量 | 376.54 |
分子式 | C18H24N4OS2< |
可溶性/溶解性 | Soluble to 75 mM in DMSO and to 10 mM in ethanol |
参考文献 | McKayet al (2012) Direct pharmacological monitoring of the developmental switch in NMDAR subunit composition using TCN 213, a GluN2A-selective, glycine-dependent antagonist. Br.J.Pharmacol. 166 924. PMID: 22022974. Bettiniet al (2010) Identification and characterization of novel NMDA receptor antagonists selective for NR2A- over NR2B-containing receptors. J.Pharmacol.Exp.Ther. 335 644. PMID: 20810618. |