货号 | 5289/50 |
别名 | 4-Bromo-N-(2,3-dihydro-6-methoxy-1, |
供应商 | Tocris |
生物活性 | Selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500 nM respectively). Exhibits 39-fold selectivity for BRPF1B and BRPF2 over BRD4. Accelerates FRAP recovery at 5 μM in a BRPF2 FRAP assay. |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >98 % |
计算分子量 | 440.31 |
分子式 | C17H18BrN3O4 |
可溶性/溶解性 | Soluble to 20 mM in DMSO |