| 货号 | 4172/50 |
| 别名 | 2-Hydroxy-4-[4-(5Z)-5-[(E)-2-methyl |
| 供应商 | Tocris |
| 生物活性 | Selective antagonist for the GPR35 orphan receptor GPCR (IC50 = 20.1 nM). Over 1000-fold more selective for GPR35 compared to GPR55 antagonists. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >98 % |
| 计算分子量 | 482.57 |
| 分子式 | C24H22N2O5 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Jenkinset al (2012) Antagonists of GPR35 display high species ortholog selectivity and varying modes of action. J.Pharmacol.Exp.Ther. 343 683. PMID: 22967846. Heynen-Genelet al (2010) Antagonists for the orphan receptor GPR35. Probe Reports from the Molecular Libraries Program NBK5070. |