| 货号 | 4756/50 |
| 别名 | N-(Adamant-1-yl)-4-oxo-1-pentyl-6-p |
| 供应商 | Tocris |
| 生物活性 | Selective inverse agonist of CB2 receptors (Ki values are 3.8 and >10,000 nM for CB2 and CB1, respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 468.63 |
| 分子式 | C31H36N2O2 |
| 可溶性/溶解性 | Soluble to 100 mM in ethanol and to 20 mM in DMSO |
| 参考文献 | Contarteseet al (2012) A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury. Pharmacol.Res. 66 555. PMID: 23036353. Pasquiniet al (2008) Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J.Med.Chem. 51 5075. PMID: 18680276. |