| 货号 | 3556/50 |
| 别名 | N-(Adamant-1-yl)-6-isopropyl-4-oxo- |
| 供应商 | Tocris |
| 生物活性 | Potent and selective CB2 receptor agonist (Ki values are 6.3 nM and 1.2 μM for CB2 and CB1 receptors respectively). Displays analgesic activity in the formalin test in mice. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 434.61 |
| 分子式 | C28H38N2O2 |
| 可溶性/溶解性 | Soluble to 25 mM in DMSO and to 50 mM in ethanol |
| 参考文献 | Contartese (2012) A novel CB2 agonist, COR167, potently protects rat brain cortical slices against OGD and reperfusion injury. Pharmacol.Res. 66 555. PMID: 23036353. Pasquiniet al (2008) Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J.Med.Chem. 51 5075. PMID: 18680276. |