货号 | 2270/50 |
别名 | 2-(2-Furanyl)-7-(2-phenylethyl)-7H- |
供应商 | Tocris |
生物活性 | Potent and selective A2A adenosine receptor competitive antagonist (Ki = 1.3 nM). Displays 323-, 53- and 100-fold selectivity over A1, A2B and A3 receptors, respectively. |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >99 % |
计算分子量 | 345.36 |
分子式 | C18H15N7O |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
CAS号 | 160098-96-4 |
参考文献 | Bastiaet al (2002) Effects of A1 and A2A adenosine receptor ligands in mouse acute models of pain. Neurosci.Lett. 328 241. PMID: 12147316. Belardinelliet al (1997) The A2A adenosine receptor mediates coronary vasodilation. J.Pharmacol.Exp.Ther. 2841066. Zocchiet al (1996) Binding of the radioligand [3H]-SCH 58261, a new non-xanthine A2A adenosine receptor antagonist, to rat striatal membranes. J.Pharmacol.Exp.Ther. 276 398. PMID: 8632302. |