| 货号 | 2993/50 |
| 别名 | 4-(4-Fluoro-1-naphthalenyl)-6-(1-me |
| 供应商 | Tocris |
| 生物活性 | High affinity 5-HT2B receptor antagonist (pKi = 9.5). Displays 1000-fold selectivity for 5-HT2B with good bioavailability. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 317.79 |
| 分子式 | C17H16FN3.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
| CAS号 | 199864-87-4 |
| 参考文献 | Callebertet al (2006) Evidence for a control of plasma serotonin levels by 5-Hydroxytryptamine2B receptors in mice. J.Pharmacol.Exp.Ther. 317 724. PMID: 16461587. Bonhauset al (1999) RS-127445: a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist. Br.J.Pharmacol. 127 1075. PMID: 10455251. |