NPS ALX Compound 4a dihydrochloride (50 MG)
货号:
3285/50 基本售价:
11381.8 元 规格:
50 mg
产品信息
概述货号 | 3285/50 |
别名 | 6-(Hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-1-(1-naphthalenylsulfonyl)-1H-indole dihydrochloride |
性能供应商 | Tocris |
生物活性 | Potent and competitive 5-HT6 antagonist (IC50 = 7.2 nM, Ki = 0.2 nM) that displays selectivity over other 5-HT and D2receptors. |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >99 % |
计算分子量 | 504.47 |
分子式 | C25H25N3O2S.2HCl |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
CAS号 | 299433-10-6 |
参考文献 | Isaacet al (2000) 6-bicyclopiperazinyl-1-arylsulfonylindoles and 6-bicyclopiperidinyl-1-arylsulfonylindoles derivatives as novel, potent, and selective 5-HT6 receptor antagonists. Bioorg.Med.Chem.Letts. 101719. |