| 货号 | 3921/50 |
| 别名 | N-(Piperidin-1-yl)-5-(4-methoxyphen |
| 供应商 | Tocris |
| 生物活性 | High affinity CB1 receptor antagonist (Ki = 4.1 nM). Exhibits significantly reduced lipophilicity compared to other CB1antagonists. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 459.37 |
| 分子式 | C23H24Cl2N4O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 100 mM in ethanol |
| CAS号 | 502486-89-7 |
| 参考文献 | Milleret al (2007) Analogs of SR-141716A (Rimonabant) alter d-amphetamine-evoked [3H] dopamine overflow from preloaded striatal slices and amphetamine-induced hyperactivity. Life Sci. 81 63. PMID: 17532007. Katoch-Rouseet al (2003) Synthesis, structure-activity relationship and evaluation of SR141716 analogues: development of central cannabinoid receptor ligands with lower lipophilicity. J.Med.Chem. 46 642. PMID: 12570386. |