| 货号 | 4878/50 |
| 别名 | (Z,Z)-4,4'-[1,3-Phenylenebis(oxy-4,1 |
| 供应商 | Tocris |
| 生物活性 | Potent and selective lysophosphatidic acid 2 (LPA2) receptor antagonist (IC50 values are 8.9, 1230 and 27354 nM for LPA2, LPA3 and LPA1 receptors respectively, in a LPA-elicited calcium mobilization assay). |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 488.45 |
| 分子式 | C26H20N2O8 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Fellset al (2009) Structure-based drug design identifies novel LPA3 antagonists. Bioorg.Med.Chem. 17 7457. PMID: 19800804. Fellset al (2008) Identification of non-lipid LPA3 antagonists by virtual screening. Bioorg.Med.Chem. 16 6207. PMID: 18467108. |