| 货号 | 3433/50 |
| 别名 | 3-[[[2-Methoxy-4-(phenylamino)pheny |
| 供应商 | Tocris |
| 生物活性 | Selective PPARδ antagonist (IC50 values are 0.155, > 10 and ≥10μM at PPARδ, PPARα and PPARγ respectively). Exhibits inverse agonist effects when administered by itself. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >99 % |
| 计算分子量 | 418.49 |
| 分子式 | C19H18N2O5S2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 10 mM in ethanol |
| CAS号 | 1014691-61-2 |
| 参考文献 | Bishop-Bailey and Swales (2008) The role of PPARs in the endothelium: Implications for cancer therapy. PPAR Res. 904851. Sheareret al (2008) Identification and characterization of a selective peroxisome proliferator-activated receptor β/δ (NR1C2) antagonist. Mol.Endocrinol. 22 523. PMID: 17975020. Wang (2008) PPAR-δ in vascular pathophysiology. PPAR Res. 164163. PMID: 19132133. |