| 货号 | 1247/50 |
| 别名 | (3-Aminopropyl)(cyclohexylmethyl)ph |
| 供应商 | Tocris |
| 生物活性 | Brain penetrant, selective GABAB receptor antagonist (IC50 = 4.9 μM). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 219.26 |
| 分子式 | C10H22NO2P |
| 可溶性/溶解性 | Soluble to 100 mM in water |
| CAS号 | 123691-14-5 |
| 参考文献 | Staubliet al (1999) GABAB receptor antagonism: facilitatory effects on memory parallel those on LTP induced by TBS but not HFS. J.Neurosci. 19 4609. PMID: 10341258. Curtis and Lacey (1998) Prolonged GABAB receptor-mediated synaptic inhibition in the cat spinal cord: an in vivo study. Exp.Brain Res. 121 319. PMID: 9746138. Froestlet al (1996) Potent, orally active GABAB receptor antagonists. Pharmacol.Rev.Comm. 8127. Lingenhoehl and Olpe (1993) Blockade of the late inhibitory postsynaptic potential in vivo by the GABAB antagonist CGP 46381. Pharmacol.Comm. 349. |