TC-E 5005 (50 MG)
货号：
4572/50 基本售价：
11233.1 元 规格：
50 mg
产品信息
概述| 货号 | 4572/50 |
| 别名 | 2-Methoxy-6,7-dimethyl-9-propyl-imidazo[1,5-a]pyrido[3,2-e]pyrazine |
性能| 供应商 | Tocris |
| 生物活性 | Potent and selective PDE10A inhibitor (IC50 values are 7.28, 239, 779, 919, 3100 and 3700 nM at PDE10A, 2A, 11A, 5A, 7B and 3A respectively and >5000 nM at PDE1B, 4A, 6, 8A and 9A). Reverses MK 801-induced hyperactivity in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >99 % |
| 计算分子量 | 270.33 |
| 分子式 | C15H18N4O |
| 可溶性/溶解性 | Soluble to 100 mM in 1eq. HCl and to 100 mM in ethanol |
| 参考文献 | Hofgenet al (2010) Discovery of imidazo[1,5-a]pyrido[3,2-e]pyrazines as a new class of phosphodiesterase 10A inhibitiors. J.Med.Chem. 53 4399. PMID: 20450197. |
