PSB 603 (50 MG)
货号:
3198/50 基本售价:
11233.1 元 规格:
50 mg
产品信息
概述货号 | 3198/50 |
别名 | 8-[4-[4-(4-Chlorophenzyl)piperazide-1-sulfonyl)phenyl]]-1-propylxanthine |
性能供应商 | Tocris |
生物活性 | Adenosine A2B receptor antagonist that displays > 17000-fold selectivity over other adenosine receptors (Ki values are 0.553, > 10000, > 10000 and > 10000 nM for A2B, A1, A2A and A3 receptors respectively). |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >98 % |
计算分子量 | 529.01 |
分子式 | C24H25ClN6O4S |
可溶性/溶解性 | Soluble to 50 mM in DMSO |
参考文献 | Borrmannet al (2009) 1-alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: development and characterization of adenosine A2B receptor antagonists and a new radioligand with subnanomolar affinity and subtype specificity. J.Med.Chem. 52 3994. PMID: 19569717. |