| 货号 | 1644/50 |
| 别名 | N'-[(8-α1,6-dimethylergolin-8-yl]-N,N |
| 供应商 | Tocris |
| 生物活性 | 5-HT2Aand2C receptor antagonist (pA2 values are 9.1 for each receptor) and D2-like dopamine receptor partial agonist (Ki = 8 nM). Displays antiprolactin and antiparkinsonian effects in vivo. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 398.95 |
| 分子式 | C18H26N4O2S.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 5 mM in water with gentle warming |
| CAS号 | 64795-35-3 |
| 参考文献 | Hoyeret al (1994) VII. International Union of Pharmacology classification of receptors for 5-hydroxytryptamine (serotonin). Pharmacol.Rev. 46 157. PMID: 7938165. Marko (1984) Dopamine agonistic potency of two novel prolactin release-inhibiting ergolines. Eur.J.Pharmacol. 101 263. PMID: 6468500. Markstei (1983) Mesulergine and its 1,20-N,N-bidemethylated metabolite interact directly with D1- and D2-receptors. Eur.J.Pharmacol. 95 101. PMID: 6230246. |