Tilfrinib (50 MG)
货号：
5579/50 基本售价：
11084.4 元 规格：
50 mg
产品信息
概述| 货号 | 5579/50 |
| 别名 | 3-(9H-Pyrido[2,3-b]indol-4-ylamino)phenol |
性能| 供应商 | Tocris |
| 生物活性 | Potent and selective breast tumor kinase (Brk, also known as tyrosine-protein kinase 6, PTK6) inhibitor (IC50 = 3.15 nM). Exhibits >1000-fold selectivity for Brk over a panel of other kinases. Inhibits proliferation of breast cancer cells in vitro. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 275.3 |
| 分子式 | C17H13N3O |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Mahmoudet al (2014) Discovery of 4-anilino α-carbolines as novel Brk inhibitors. Bioorg.Med.Chem.Lett. 24 1948. PMID: 24650640. |
