| 货号 | 2493/50 |
| 别名 | 4-[3-(1H-Imidazol-4-yl)propyl]piper |
| 供应商 | Tocris |
| 生物活性 | Potent histamine H3 receptor silent antagonist (pKi = 8.35). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 355.11 |
| 分子式 | C11H19N3.2HBr |
| 可溶性/溶解性 | Soluble to 100 mM in water and to 100 mM in DMSO |
| 参考文献 | Moreno-Delgadoet al (2006) Constitutive activity of H3 autoreceptors modulates histamine synthesis in rat brain through the cAMP/PKA pathway. Neuropharmacology 51 517. PMID: 16769092. Leurset al (2005) The histamine H3 receptor: from gene cloning to H3 receptor drugs. Nat.Rev.Drug Discov. 4 107. PMID: 15665857. Kitbunnadajet al (2004) Identification of 4-(1H-imidazol-4(5)-ylmethyl)pyridine (immethridine) as a novel, potent, and highly selective histamine H3 receptor agonist. J.Med.Chem. 47 2414. PMID: 15115383. |