U 90042 (50 MG)
货号：
2733/50 基本售价：
10549.0 元 规格：
50 mg
产品信息
概述| 货号 | 2733/50 |
| 别名 | 11-Chloro-5-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-2,3-dihydrodiimidazo[1,5-a:1',2'-c]quinazoline |
性能| 供应商 | Tocris |
| 生物活性 | GABAA receptor ligand that binds with comparable affinities to three receptor subtypes: α1β2γ2,α3β2γ2andα6β2γ2(Ki values are 7.8, 9.5 and 11.0 nM respectively). Potentiates GABA-induced chloride currents in α6β2γ2 receptors. Sedative/hypnotic compound. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 352.78 |
| 分子式 | C17H13ClN6O |
| 可溶性/溶解性 | Soluble to 30 mM in DMSO and to 5 mM in ethanol |
| CAS号 | 134516-99-7 |
| 参考文献 | Tanget al (1995) U-90042, a sedative/hypnotic compound that interacts differentially with the GABAA receptor subtypes. J.Pharmacol.Exp.Ther. 275 761. PMID: 7473164. |
