TTP 22 (50 MG)
货号:
4432/50 基本售价:
10549.0 元 规格:
50 mg
产品信息
概述货号 | 4432/50 |
别名 | 3-[[5-(4-Methylphenyl)thieno[2,3-d]pyrimidin-4-yl]thio]propanoic acid |
性能供应商 | Tocris |
生物活性 | High affinity, ATP-competitive casein kinase 2 (CK2) inhibitor (IC50 = 0.1 μM, Ki = 40 nM). Displays selectivity for CK2 over JNK3, ROCK1 and MET (no inhibitory effects at 10 μM). |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >98 % |
计算分子量 | 330.42 |
分子式 | C16H14N2O2 |
可溶性/溶解性 | Soluble to 100 mM in DMSO and to 20 mM in ethanol |
参考文献 | Golubet al (2011) Synthesis and biological evaluation of substituted (thieno[2,3-d]pyrimidin-4-ylthio)carboxylic acids as inhibitors of human protein kinase CK2. Eur.J.Med.Chem. 46 870. PMID: 21276643. |