| 货号 | 0379/50 |
| 别名 | 3-Aminopropyl(methyl)phosphinic acid; CGP 35024 |
| 供应商 | Tocris |
| 生物活性 | Very potent GABAB agonist, at least ten times more active than baclofen (Cat. No. 0417). Also GABAA-ρantagonist. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 计算分子量 | 137.12 |
| 分子式 | C4H12NO2P |
| 可溶性/溶解性 | Soluble to 100 mM in water |
| CAS号 | 127729-35-5 |
| 参考文献 | Bon and Galvan (1996) Electrophysiological characterization of GABAB agonists and antagonists in dorso-lateral septal neurones in vitro. Br.J.Pharmacol. 118 961. PMID: 8799569. Johnston (1996) GABAC receptors: relatively simple transmitter-gated ion channels? TiPS 17 319. PMID: 8885697. Froestlet al (1995) Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists. J.Med.Chem. 38 3297. PMID: 7650684. Seabrooket al (1990) Electrophysiological characterization of potent agonists and antagonists on pre- and postsynaptic GABAB receptors on neurones in brain slices. Br.J.Pharmacol. 101 949. PMID: 1964824. |