| 货号 | 1206/50 |
| 别名 | 8-Chloro-dibenzo(Z)[b,f][1,4]oxazep |
| 供应商 | Tocris |
| 生物活性 | Selective EP1 receptor antagonist (IC50 = 6.7 μM for inhibition of [3H]-PGE2 binding to EP1 transfected COS cells). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 331.76 |
| 分子式 | C16H14ClN3O3 |
| 可溶性/溶解性 | Soluble to 25 mM in ethanol with gentle warming and to 100 mM in DMSO |
| CAS号 | 19395-87-0 |
| 参考文献 | Botellaet al (1995) Receptor subtypes involved in dual effects induced by prostaglandin E2 in circular smooth muscle from dog colon. J.Pharmacol.Exp.Ther. 273 1008. PMID: 7791070. Funket al (1993) Cloning and expression of a cDNA for the human prostaglandin E receptor EP1 subtype. J.Biol.Chem. 268 26767. PMID: 8253813. Sanner (1972) Dibenzoxazepine hydrazides as prostaglandin antagonists. Intra-Science Chem.Rept. 61. |