| 货号 | 3983/50 |
| 别名 | 1-Amino-9,10-dihydro-9,10-dioxo-4-[ |
| 供应商 | Tocris |
| 生物活性 | Highly potent P2Y12 receptor antagonist (Ki = 24.9 nM). Unlike clopidogrel (Cat. No. 2490), does not require bioactivation. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >95 % |
| 计算分子量 | 609.54 |
| 分子式 | C26H17N3Na2< |
| 可溶性/溶解性 | Soluble to 25 mM in water |
| 参考文献 | Felixet al (2011) Development of a comprehensive set of P2 receptor pharmacological research compounds. Purinerg.Sig. 8 101. PMID: 22052555. Baqiet al (2009) High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12 receptors. J.Med.Chem. 52 3784. PMID: 19463000. Hoffmannet al (2009) Interaction of new, very potent non-nucleotide antagonists with Arg256 of the human platelet P2Y12 receptor. J.Pharmacol.Exp.Ther. 331 648. PMID: 19690189. |