SDM25N hydrochloride (50 MG)
货号:
1410/50 基本售价:
10489.5 元 规格:
50 mg
产品信息
概述货号 | 1410/50 |
别名 | (4bS,8R,8aS,14bR)-5,6,7,8,14,14b-Hexahydro-7-(2-methyl-2-propenyl)-4,8-methanobenzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol hydrochloride |
性能供应商 | Tocris |
生物活性 | Potent and highly selective non-peptide δ receptor antagonist (Ki values are 4.7, 3800 and 7900 nM for δ,κandμ receptors respectively). More selective than naltrindole (Cat. No. 0740). |
运输条件 | Blue Ice |
存放说明 | 4℃ |
纯度 | >99 % |
计算分子量 | 450.96 |
分子式 | C26H26N2O3.HCl |
可溶性/溶解性 | Soluble to 10 mM in water and to 100 mM in DMSO |
CAS号 | 342884-62-2 |
参考文献 | McLamoreet al (2001) Effect of N-alkyl and N-alkenyl substituents in noroxymorphindole, 17-substituted-6,7-dehydro-4,5α-epoxy-3,14-dihydroxy-6,7:2 ',3 '-indolomorphinans, on opioid receptor affinity, selectivity, and efficacy. J.Med.Chem. 44 1471. PMID: 11311071. |