| 货号 | 0899/50 |
| 别名 | 7-Benzylidenenaltrexone maleate |
| 供应商 | Tocris |
| 生物活性 | Standard selective δ1 opioid receptor antagonist. Also inhibits neurogenic ion transport mediated by a putative novel opioid receptor in porcine ileal mucosa. |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 纯度 | >99 % |
| 计算分子量 | 545.59 |
| 分子式 | C27H27NO4.C4H4O4 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 10 mM in water with gentle warming |
| CAS号 | 129468-28-6 |
| 参考文献 | Poonyachotiet al (2001) Pharmacological evidence for a 7-benzylidenenaltrexone-preferring opioid receptor mediating the inhibitory actions of peptidic δ- and μ-opioid agonists on neurogenic ion transport in porcine ileal mucosa. J.Pharmacol.Exp.Ther. 297 672. PMID: 11303057. Hammondet al (1995) Antinociception and d-1 opioid receptors in the rat spinal cord: studies with intrathecal 7-benzylidenenaltrexone. J.Pharmacol.Exp.Ther. 274 1317. PMID: 7562504. Portogheseet al (1992) A δ1-opioid receptor antagonist: 7-benzylidenenaltrexone. Eur.J.Pharmacol. 218 195. PMID: 1327826. |