货号 | 1385/50 |
别名 | 1,4-Dihydro-2-methyl-6-phenyl-4-(ph |
供应商 | Tocris |
生物活性 | Potent and highly selective antagonist for the human adenosine A3 receptor. Ki values are 2.69 nM at hA3, and > 100 μM at rat A1 and rat A2Areceptors. |
运输条件 | Blue Ice |
存放说明 | -20℃ |
纯度 | >98 % |
计算分子量 | 522.56 |
分子式 | C31H26N2O6 |
可溶性/溶解性 | Soluble to 100 mM in DMSO |
CAS号 | 192053-05-7 |
参考文献 | Baraldi and Borea (2000) New potent and selective human adenosine A3 receptor antagonists. TiPS 21 456. PMID: 11121831. Liet al (1998) Structure-activity relationships and molecular modeling of 3,5-diacyl-2,4-dialkylpyridine derivatives as selective A3 adenosine receptor antagonists. J.Med.Chem. 41 3186. PMID: 9703464. |