| 货号 | 0779/50 |
| 别名 | N-[2-(4-Iodophenyl)ethyl]-S-[3-(4(5 |
| 供应商 | Tocris |
| 生物活性 | Selective H3 antagonist with high affinity (KD = 0.3 nM). Also available as part of the Histamine H3 Receptor Tocriset™. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 576.13 |
| 分子式 | C15H19IN4S.2HBr |
| 可溶性/溶解性 | Soluble to 25 mM in water |
| CAS号 | 143407-29-8 |
| 参考文献 | Shahidet al (2009) Histamine, histamine receptors, and their role in immunomodulation: An updated systematic review. Open Immunol.J. 29. Jansenet al (1994) Characterisation of the binding of the first selective radiolabelled histamine H3 receptor antagonist, [125I]-iodophenpropit, to rat brain. Br.J.Pharmacol. 113 355. PMID: 7834183. Jansenet al (1992) The first radiolabelled histamine H3 receptor antagonist, [125I]iodophenpropit: saturable and reversible binding to rat cortex membranes. Eur.J.Pharmacol. 217 203. PMID: 1330590. Mengeet al (1992) Synthesis of S-[3-(4(5)-imidazolyl)propyl]-N-[2-(4-[125I]-iodophenylethyl]isothiourea sulfate [125I]-iodophenpropit), a new probe for histamine H3 receptor binding sites. J.Labelled Comp.Radiopharm. XXXI 10781. |