CYM 5541 (50 MG)
货号：
4897/50 基本售价：
10192.1 元 规格：
50 mg
产品信息
概述| 货号 | 4897/50 |
| 别名 | N,N-Dicyclohexyl-5-cyclopropyl-3-isoxazolecarboxamide |
性能| 供应商 | Tocris |
| 生物活性 | Selective sphingosine-1-phosphate receptor 3 (S1P3) allosteric agonist (EC50 = 72-132 nM). Occupies a different space within the ligand binding pocket of S1P3 than S1P. Displays no activity at S1P1, S1P2, S1P4 and S1P5 receptors at concentrations up to 10 μM. Shows no significant activities in a profiling panel of 55 GPCRs, ion channels and transporters. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >97 % |
| 计算分子量 | 316.44 |
| 分子式 | C19H28N2O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 50 mM in ethanol |
| 参考文献 | Joet al (2012) Novel selective allosteric and bitopic ligands for the S1P3 receptor. ACS Chem.Biol. 7 1975. PMID: 22971058. |
