TCS PIM-1 1 (50 MG)
货号：
2979/50 基本售价：
9894.7 元 规格：
50 mg
产品信息
概述| 货号 | 2979/50 |
| 别名 | 3-Cyano-4-phenyl-6-(3-bromo-6-hydroxy)phenyl-2(1H)-pyridone |
性能| 供应商 | Tocris |
| 生物活性 | ATP-competitive Pim-1 kinase inhibitor that displays selectivity over Pim-2 and MEK1/2 (IC50 values are 50, > 20000 and > 20000 nM for Pim-1, Pim-2 and MEK1/2 respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 367.2 |
| 分子式 | C18H11BrN2O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| 参考文献 | Cheneyet al (2007) Identification and structure-activity relationships of substituted pyridones as inhibitors of Pim-1 kinase. Bioorg.Med.Chem.Letts. 17 1679. PMID: 17251021. |
