TCS 1105 (50 MG)
货号：
3942/50 基本售价：
9894.7 元 规格：
50 mg
产品信息
概述| 货号 | 3942/50 |
| 别名 | N-[(-4-Fluorophenyl)methyl]-α-oxo-1H-indole-3-acetamide |
性能| 供应商 | Tocris |
| 生物活性 | GABAA benzodiazepine receptor (BZR) ligand. Acts as an agonist at α2 and antagonist at α1 benzodiazepine receptors (Ki values are 118 and 245 nM respectively). Anxiolytic agent lacking sedative activity. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 296.3 |
| 分子式 | C17H13FN2O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO and to 20 mM in ethanol |
| CAS号 | 185391-33-7 |
| 参考文献 | Talianiet al (2009) Identification of anxiolytic/nonsedative agents among indol-3-ylglyoxylamides acting as functionally selective agonists at the γ-aminobutyric acid-A (GABAA) α2 benzodiazepine receptor. J.Med.Chem 52 3723. PMID: 19469479. |
