| 货号 | 1991/50 |
| 别名 | 1,3-Bis(4-hydroxyphenyl)-4-methyl-5 |
| 供应商 | Tocris |
| 生物活性 | Selective, high affinity silent antagonist at ERα receptors. Displays > 200-fold selectivity for ERα over ERβ. Ki values are 2.7 and 1800 nM at ERα and ERβ receptors respectively. |
| 运输条件 | Blue Ice |
| 存放说明 | 4℃ |
| 纯度 | >98 % |
| 计算分子量 | 542.5 |
| 分子式 | C29H31N3O3.2HCl |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| CAS号 | 289726-02-9 |
| 参考文献 | Harringtonet al (2003) Activities of estrogen receptor alpha- and beta-selective ligands at diverse responsive gene sites mediating transactivation or transrepression. Mol.Cell.Endocrinol. 206 13. PMID: 12943986. Sunet al (2002) Antagonists selective for estrogen receptor α. Endocrinol. 143941. |