| 货号 | 1018/50 |
| 别名 | 2-[2-(5-Bromo-1H-indol-3-yl)ethyl]- |
| 供应商 | Tocris |
| 生物活性 | Potent CCK2 receptor antagonist (IC50 = 9.3 nM for inhibition of 125I-labeled CCK-8 sulfate binding at mouse brain membranes). |
| 运输条件 | Blue Ice |
| 存放说明 | -20℃ |
| 计算分子量 | 502.41 |
| 分子式 | C27H24BrN3O2 |
| 可溶性/溶解性 | Soluble to 100 mM in DMSO |
| CAS号 | 133040-77-4 |
| 参考文献 | Suman-Chauhanet al (1996) The influence of guanyl nucleotide on agonist and antagonist affinity at guinea-pig CCK-B / gastrin receptors: binding studies using [3H]PD140376. Regul.Pept. 65 37. PMID: 8876034. Yuet al (1991) Quinazolinone cholecystokinin receptor ligands. J.Med.Chem. 34 1505. PMID: 2016728. |