| 货号 | 1357/50 |
| 别名 | 2,3-Dihydro-5,6-dimethoxy-N,N-dipropyl-1H-inden-2-amine maleate; PNU 99194 |
| 供应商 | Tocris |
| 生物活性 | Potent, selective D3 antagonist. Ki values are 160, 2281 and > 10000 nM for human cloned D3, D2 and D4 receptors respectively. |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 393.48 |
| 分子式 | C17H27NO2.C4H4O4 |
| 可溶性/溶解性 | Soluble to 25 mM in water |
| CAS号 | 83598-46-3 |
| 参考文献 | LaHosteet al (2000) Dopamine D1 receptors synergize with D2, but not D3 or D4, receptors in the striatum without the involvement of action potentials. J.Neurosci. 20 6666. PMID: 10964971. Audinotet al (1998) A comparative in vitroandin vivo pharmacological characterization of the novel dopamine D3 receptor antagonists (+)-S 14297, nafadotride, GR 103,691 and U 99194. J.Pharmacol.Exp.Ther. 287 187. PMID: 9765337. Clifford and Waddington (1998) Heterogeneity of behavioural profile between three putative selective D3 dopamine receptor antagonists using an ethologically based approach. Psychopharmacology 136 284. PMID: 9566814. |