| 货号 | 2034/50 |
| 别名 | N-[3-(1H-Imidazol-4-yl)propyl]-1H-b |
| 供应商 | Tocris |
| 生物活性 | Potent H3 antagonist (pKB at guinea-pig ileum H3-receptor = 9.46). Limited blood brain barrier permeability (ED50 = 19.12 mg/kg i.p.). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >99 % |
| 计算分子量 | 421.37 |
| 分子式 | C13H15N5.2C2H2O4 |
| 可溶性/溶解性 | Soluble to 50 mM in water and to 50 mM in DMSO |
| CAS号 | 184576-87-2 |
| 参考文献 | Moret al (2004) Synthesis, biological activity, QSAR and QSPR study of 2-aminobenzimidazole derivatives as potent H3-antagonists. Bioorg.Med.Chem.Lett. 12663. Ballabeniet al (2002) CNS access of selected H3-antagonists: ex vivo binding study in rats. Inflamm.Res. 51 (Suppl 1) S55. PMID: 12013409. |