NS 3763 (50 MG)
货号:
2187/50 基本售价:
8704.9 元 规格:
50 mg
产品信息
概述货号 | 2187/50 |
别名 | 4,6-Bis(benzoylamino)-1,3-benzenedicarboxylic acid |
性能供应商 | Tocris |
生物活性 | Selective non-competitive kainate receptor antagonist; displays selectivity for GLUK5 subunit-containing receptors (IC50 values are 1.6 and > 30 μM for homomeric GLUK5 and GLUK6 receptors respectively). Has minimal activity at AMPA and NMDA receptors (IC50> 30 μM). |
运输条件 | Blue Ice |
存放说明 | Ambient |
纯度 | >98 % |
计算分子量 | 404.38 |
分子式 | C22H16N2O6 |
可溶性/溶解性 | Soluble to 25 mM in DMSO |
CAS号 | 70553-45-6 |
参考文献 | Christensenet al (2004) In vitro characterization of 5-carboxyl-2,4-di-benzamido-benzoic acid (NS3763), a noncompetitive antagonist of GLUK5 receptors. J.Pharmacol.Exp.Ther. 309 1003. PMID: 14985418. |