| 货号 | 0793/50 |
| 别名 | 2-(1,4-Benzodioxan-2-yl)-2-imidazol |
| 供应商 | Tocris |
| 生物活性 | α2-adrenoceptor antagonist, and I2 ligand, selective over I1 sites (pKi values are 5.90, 7.22, 8.01, 7.43, and 7.7 for I1, I2,α2A,α2B, and α2C receptors respectively). |
| 运输条件 | Blue Ice |
| 存放说明 | Ambient |
| 纯度 | >98 % |
| 计算分子量 | 240.69 |
| 分子式 | C11H12N2O2.HCl |
| 可溶性/溶解性 | Soluble to 100 mM in water |
| CAS号 | 79944-56-2 |
| 参考文献 | Eglenet al (1998) 'Seeing through a glass darkly': casting light on imidazoline 'I' sites. TiPS 19 381. PMID: 9786027. Berdeuet al (1995) Evidence for two different imidazoline sites on pancreatic B cells and vascular bed in rat. Eur.J.Pharmacol. 275 91. PMID: 7774667. Michel and Ernsberger (1992) Keeping an eye on the I site: imidazoline-preferring receptors. TIPS 13 369. PMID: 1413085. Dabir (1986) Idazoxan: a novel pharmacological tool for the study of α2-adrenoceptors. J.Pharmacol. 17 113. PMID: 2875218. |